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The details of the synthetic sequence followed for the preparation of all these compounds having almost all the structural features required for a compound to act as a potent insulin sensitizing agent are reported.
      
Both these models predicted binding affinity of internal and external test set compounds including the enantiomers of compound no.
      
Aminochalcone 18, which has an IC50 value of 0.24 μM, was the most potent compound.
      
When tested on a wide battery of receptors, including 5HT2A(h), 5HT3(h), α1, α 2, β1, β2, H1, H2, opioids, D1(h), D2(h), 5HT uptake, and DOPA uptake, compound 9 showed submicromolar affinity only for α2 (Ki = 205 nM) and H1 (Ki = 311 nM).
      
We designed an isatin lead compound as a novel non-nucleoside reverse transcriptase inhibitor with broad-spectrum chemotherapeutic properties for the effective treatment of AIDS and AIDS-related opportunistic infections.
      
The compound 12 was found to be five times more potent than 11 in reducing twitch response to nerve stimulations, indicating the importance of extended interonium distances and 17-acetoxy function for potent antagonist activity.
      
Compound 4b exhibited bactericidal activity agains S.
      
While compound 8a showed distinct antifungal activity against C.
      
While compound 28 proved to be potent against Salmonella typhi and Klebsiella pneumoniae.
      
Finally, we applied the model for prediction of a promising new BABQ compound expected to be highly active, and it is seen that our model is in good agreement with the hypothesis in terms of in vitro and in vivo activities.
      
Compound 6 exerted potent in vitro antibacterial activity against B.
      
subtilis while compound 6 exhibited in vitro antifungal activity against Candida-6.
      
Indeed, compound 13c showed the highest activity profile against individual leukemia subpanel cell line SR (GI50?=?0.91?μM).
      
Compound IVa showed the best antifungal activity compared with miconazole (CAS 22916-47-8).
      
Compound IVc indicated the best antibacterial activity compared with the control drug ampicillin (CAS 69-53-4).
      
Compound 1-benzhydryl-4-(4-tert-butyl-benzenesulfonyl)-piperazine (7d) showed significant inhibitory activity.
      
Compound 4, 5, 6, 7, and 8 were synthesized from 4-benzoyl-1,5-diphenyl-1H-pyrazole-3-carboxylic acid 1 as a starting material.
      
The finding of antibacterial activity study showed that the sulfamide derivative 5 was the best compound of the series, exhibiting antibacterial activity against both Gram-positive and Gram-negative bacteria.
      
Both infrared spectra and melting point of the compound were consistent with those reported earlier.
      
Analytical results for two batches of compound ibuprofen tablets by the SEKI-based FI-CE approach were in good agreement with that obtained by a conventional high performance liquid chromatographic method.
      
 

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